Owner Arena Pharmaceuticals, Inc.

Inventors Jones, Robert M.; Han, Sangdon; Thoresen, Lars; Jung, Jae-Kyu; StrahPleynet, Sonja; Zhu, Xiuwen; Xiong, Yifeng; Yue, Dawei

Agent FB Rice

Pub. Number AU-A-2010286988

PCT Pub. Number WO2011/025541

Priority 61/275,506 28.08.09 US; 61/400,146 22.07.10 US; 61/396,588 28.05.10 US

Filing date 27 August 2010

Wipo publication date 3 March 2011

C07D 231/54 (2006.01) Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings

A61K 31/416 (2006.01) - condensed with carbocyclic ring systems, e.g. indazole

A61K 31/4439 (2006.01)

A61K 31/497 (2006.01)

A61K 31/661 (2006.01) - Phosphorus acids or esters thereof not having PC bonds, e.g. fosfosal, dichlorvos, malathion

A61P 19/02 (2006.01) Drugs for skeletal disorders

A61P 29/00 (2006.01) Non-central analgesic, antipyretic or antiinflammatory agents, e.g antirheumatic agents

C07D 401/04 (2006.01) Heterocyclic compounds containing two or more hetero rings

C07D 401/14 (2006.01) Heterocyclic compounds containing two or more hetero rings

C07D 403/04 (2006.01) Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group

C07D 405/14 (2006.01) Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom

C07F 9/09 (2006.01) Compounds containing elements of the 5th Group of the Periodic System