Owner Merck Sharp & Dohme Corp.

Inventors Isaacs, Richard C. A.; Thompson, Wayne J.; Williams, Peter D.; Su, DaiShi; Venkatraman, Shankar; Embrey, Mark W.; Fisher, Thorsten E.; Wai, John S.; Dubost, David C.; Ball, Richard G.; Choi, Eric J.; Pei, Tao; Trice, Sarah L.; Campbell, Neil; Maddess, Matthew; Maligres, Peter E.; Shevlin, Michael; Song, Zhiguo Jake; Steinhuebel, Dietrich P.; Strotman, Neil A.; Yin, Jingjun

Agent Spruson & Ferguson

Pub. Number AU-A-2009302663

PCT Pub. Number WO2010/042392

Priority 61/195,271 06.10.08 US

Filing date 2 October 2009

Wipo publication date 15 April 2010

C07D 281/10 (2006.01) Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms

A61K 31/55 (2006.01) - having seven-membered rings, e.g. azelastine, pentylenetetrazole

A61K 31/553 (2006.01) - having at least one nitrogen and at least one oxygen as ring hetero atoms, e.g. loxapine, staurosporine

A61P 31/18 (2006.01) Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics

C07D 487/04 (2006.01) Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups